I-PKC ne-ROCK

I-AR-13324 hydrochloride yi-ROCK, futhi i-norepinephrine transporter inhibitor.AR-13324 Hydrochloride (i-Netarsudil) i-Rho kinase inhibitor ene ...

I-AR-13324 iyi-inhibitor encane ye-Rho kinase ne-norepinephrine transporter; kuncishisa ukucindezelwa kwe-intraocular (IOP) ku-normotensive mon ...

Enzastaurin (LY317615) lungumbulali PKCβ inhibitor abakhethayo nge IC50 ka 6 nm, 6 kuya selectivity 20-nesibaya ngokumelene PKCα, PKCγ futhi PKCε ....

I-Fasudil Hcl (HA-1077; AT-877) iyinhibitha enamandla ka-ROCK-II, PKA, PKG, PKC, ne-MLCK nge-Ki ye-0.33 μM, i-1.6 μM, i-1.6 μM, i-3.3 μM ne-36 μM, ...

I-Bisindolylmaleimide I (GF109203X) iyi-inhibitor yeprotheyini kinase C (PKC) ekhethiwe kakhulu, ebonakalayo, futhi eguquguqukayo ne-Ki Ki ye-1 ...

Hamba i-6983 i-pan-PKC inhibitor ephikisana no-PKCα, PKCβ, PKCγ ne-PKCδ nge -IC50 ye-7 nM, i-7 nM, i-6 nM ne-10 nM, ngokulandelana; Kunamandla kakhulu ku-PKC ...

I-GSK269962A (GSK269962) iyinhlangano enamandla ye-ROCK inhibitor (amanani we-IC50 ayi-1.6 no-4 nM we-ROCK1 wabantu abasha kanye ne-ROCK2 ngokulandelanayo); ibonisa ...

Isizinda samahhala se-Ripasudil (isisekelo samahhala se-K-115) siyisimangalo esithile se-ROCK, nama-IC50 we-19 no-51 nM we-ROCK2 no-ROCK1, ngokulandelana ....

I-KD025 iyatholakala ngomlomo, futhi i-ROCK2 inhibitor ene-IC50 ne-Ki ye-60nM ne-41 nM, ngokulandelana ...

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LX7101 kuyinto inhibitor elinamandla LIMK futhi ROCK2 nge IC50 namagugu 24, 1.6 futhi 10 nm ngoba LIMK1, LIMK2 futhi ROCK2, ngokulandelana; futhi inhibits ...

I-LY411575 iyinhlangano enamandla kakhulu ye-γ-secretase inhibitor ene-IC50 ye-0.078 nM / 0.082 nM (i-membrane / cell-based-based), futhi ivimba ukuchithwa kwe-Notch nge -IC50 ye ...

I-MK-0752 i-γ-secretase inhibitor enamandla kakhulu, ehlisa ukukhiqizwa kwe-Aβ40 ne-IC50 ye-5 nM. Isigaba 1 / 2 ....

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