Uke wazibuza ukuthi kusho ukuthini uma uya esitolo bese ubheka al.

Ukubonisa 1-12 of 29 imiphumela

I-CAS CHA. I-PRODUCT NAME ISENDLALELO
    1527503-11-2 A-366 (1527503-11-2)

    A-366 yi-G9a / GLP i-histone lysine methyltransferase inhibitor enamandla futhi ekhethiwe (IC₅₀ = 3.3 nM). Ikhombisa> ukukhetha kwe-1000-fold for ...

    328968-36-1 I-C646 (328968-36-1)

    I-C646 iyinhibitha ye-histone acetyltransferase, futhi ivimbela i-p300 nge-Ki ye-400 nM. Okukhethayo ngokukhetha i-p300 ngokumelene nezinye i-ace ...

    1163-36-6 I-Clemizole HCL (i-1163-36-6)

    I-Clemizole hydrochloride yi-H1 i-histamine receptor antagonist, itholakala ekuvimbela kakhulu ukuphindaphinda kwe-HCV. I-IC50 ye-Clemizole ...

    1621862-70-1 I-CPI-1205 (1621862-70-1)

    I-CPI-1205 iyinhibitha ye-histone lysine methyltransferase e-EZH2, ene-potentially antinoplastic activity.

    ...
    1396772-26-1 EPZ005687 (1396772-26-1)

    I-EPZ005687 iyi-inhibitor enamandla futhi ekhethiwe ye-EZH2 ne-Ki ye-24 nM, ukukhethwa kwe-50 ngokumelene no-EZH1 kanye ne-500-fold selectivity ngokumelene ne-15 ...

    1616391-65-1 EPZ015666 (1616391-65-1)

    I-EPZ015666 iyinhlangano enamandla yokukhetha i-PRMT5 inhibitor (Ki ka-5 nM); ukubonisa> ukukhethwa kwe-20,000 ngokulandelana kwamanye ama-PMT. I-EPZ015666 yenza nge-blocki ...

    1616391-87-7 EPZ015866 (GSK591) (1616391-87-7)

    I-EPZ015866 (GSK591) iyinhlangano ye-arginine methyltransferase eyinhloko ye-arginine methyltransferase PRMT5 / MEP50 eyinkimbinkimbi ngaleyo ndlela ibeka i-methylation yayo ...

    1700663-41-7 EPZ020411 (1700663-41-7)

    I-EPZ020411 iyi-inhibitor enamandla futhi ekhethiwe ye-PRMT6 ne-IC50 ye-10 nM, ine> 10 ukukhetha okukhethiwe ku-PRMT6 ngaphezu kwe-PRMT1 no-PRMT8.

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    1380288-87-8 EPZ5676 (1380288-87-8)

    I-Pinometostat, eyaziwa nangokuthi i-EPZ-5676. I-Pinometostat isetshenziswe ekuhlolweni kokutadisha ukwelashwa kwe-Leukemia, i-Acute Leukemias, i-Acute Myeloid ...

    1403254-99-8 EPZ6438 (1403254-99-8)

    I-Tazemetostat (i-EPZ-6438) iyinhlangano ye-EZH2 enamandla, ekhethiwe futhi ekhona ngomlomo. UTazemetostat usetshenziswe ekuhlolweni kokutadisha ukwelashwa ...

    1373423-53-0 I-GSK J4 (1373423-53-0)

    I-GSK-J4 isetshenziselwe ukutadisha umphumela we-KDM2B (i-Jumonji (JmjC) domain histone 3 i-lysine 36 (H3K36) i-di-demethylase) inhibition ekusindeni ...

    1431368-48-7 GSK-LSD1 2HCl (1431368-48-7)

    I-GSK-LSD1 isetshenziswe njenge-lysine ethile ye-demethylase i-1 (LSD1) inhibitor kumagundane ukuze afunde ukufa kwe-sepsis-okubangelwa ukufa. Kuye kwasetshenziselwa ...