Ukubonisa 1-12 of 36 imiphumela

I-CAS CHA. I-PRODUCT NAME ISENDLALELO
    856925-71-8 (-) - iBlebbistatin (856925-71-8)

    (-) - I-Blebbistatin iyi-inhibitor yeselula engenawo umzimba i-myosin II ATPase ne-IC50 ye- ~ 2 μM, ayivimbeli i-myosin light chain kinase ...

    1268524-70-4 (+) - JQ1 (1268524-70-4)

    (+) - I-JQ1 iyinhibitha ye-BET bromodomain, ne-IC50 ye-77 nM / 33 nM ye-BRD4 (1 / 2), ebophezela kubo bonke ama-bromodomains omndeni we-BET, kodwa hhayi ukuze i-brom ...

    659730-32-2 I-AMG517 (659730-32-2)

    I-AMG 517 ingumphikisi onamandla we-TRPV1, ophikisana ne-capsaicin, i-proton, nokushisa kwe-TRPV1 nge-IC50 ye-0.76 nM, i-0.62 nM ...

    401900-40-1 I-Andarine (i-401900-40-1)

    I-Andarine iyi-reception (AR) ye-agonist ne-Ki ye-4 nM, i-selectic-selective for organ anabolic ....

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    1233339-22-4 I-AZ20 (1233339-22-4)

    I-AZ20 iyinhlangano enomlando ne-inhibitor ekhethiwe ye-ATR kinase ne-IC50 ye-5 nM, ukukhethwa kwe-8 ngokuphindaphindiwe kwe-MTOR. I-AZ20 iyinhlangano ye-ATR protein kinase i ...

    1821428-35-6 I-AZD0156 (1821428-35-6)

    I-AZD0156 iyi-ATM kinase inhibitor esemlomo, enamandla futhi ekhethiwe, evimbela umsebenzi we-kinase we-ATM kanye ne-ATM-mediated signaling, okuvimbela i-D ...

    1240299-33-5 I-AZD3514 (1240299-33-5)

    I-AZD3514 i-downregulator ye-receptor enamandla neyomlomo kanye ne-Ki ye-2.2 μMand inekhono lokunciphisa i-AR protein expression ...

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    1035270-39-3 I-AZD4547 (1035270-39-3)

    I-AZD4547 iyonaveli ekhetha i-FGFR inhibitor eqondisa i-FGFR1 / 2 / 3 nge-IC50 ye-0.2 nM / 2.5 nM / 1.8 nM, umsebenzi obuthakathaka olwa FGFR4, VEGFR2 (KDR) ...

    1352226-88-0 I-AZD6738 (1352226-88-0)

    I-AZD6738 iyinhlangano enamandla yokukhetha i-ATR inhibitor yomlomo. Kungavimbela i-ATR substrate i-Chk1 Ser345 i-phosphorylation kumaseli anenani le-IC50 le-74 ...

    860352-01-8 I-AZD7762 (860352-01-8)

    I-AZD7762 iyinhibitha enamandla futhi ekhethiwe ye-Chk1 ne-IC50 ye-5 nM. Ilingana kakhulu ne-Chk2 futhi encane kakhulu ngokumelene ne-CAM, Yebo, Fy ...

    847499-27-8 I-CEP-18770 (Delanzomib) (847499-27-8)

    I-CEP-18770 iyi-inhibitor yomlomo yomsebenzi we-chymotrypsin-like proteasome ne-IC50 ye-3.8 nM, enezingqinamba kuphela zokuvimbela ...

    905973-89-9 I-CGK733 (905973-89-9)

    I-CGK 733 iyi-inhibitor enamandla futhi ekhethiwe ye-ATM / ATR ne-IC50 ye ~ ~ 200 nM. I-CGK733 iyi-inhibitor ye-ATM ne-ATR inhibitor, ephawulekayo ...